Isoxazolo[4,5-c]pyridin-3-amine finds significant application in the field of medicinal chemistry, particularly in the development of pharmaceutical compounds. It serves as a key intermediate or building block in the synthesis of various biologically active molecules. Its structure is often utilized in the design of drugs targeting neurological disorders, such as anxiety, depression, and epilepsy, due to its ability to interact with specific receptors in the brain. Additionally, it is explored for its potential in creating anti-inflammatory and antimicrobial agents, contributing to the treatment of infections and inflammatory conditions. Researchers also investigate its role in developing kinase inhibitors, which are crucial in cancer therapy, as they can interfere with the growth and proliferation of cancer cells.