Isosteviol is widely studied for its potential therapeutic applications in the pharmaceutical industry. It exhibits anti-inflammatory, antihypertensive, and antidiabetic properties, making it a candidate for drug development targeting metabolic and cardiovascular diseases. Research shows it can modulate insulin secretion and improve glucose uptake, suggesting use in managing type 2 diabetes. It also demonstrates cardioprotective effects by helping regulate blood pressure and reduce oxidative stress in vascular tissues. In addition to medical uses, isosteviol serves as a natural sweetener and flavor modifier in the food industry, though less sweet than stevia derivatives. Its derivatives are explored as building blocks in organic synthesis due to their rigid diterpenoid structure, useful in designing new bioactive compounds. It is also investigated for antimicrobial activity and potential use in agricultural chemicals as a natural plant growth regulator.