Dehydroglyasperin C is primarily studied for its potent biological activities, particularly its anti-inflammatory and antioxidant effects. It has shown promise in inhibiting pathways involved in chronic inflammation, making it a candidate for research in inflammatory diseases such as arthritis and inflammatory bowel disease.

It also exhibits neuroprotective properties, with studies suggesting it may help protect brain cells from oxidative stress and reduce the risk of neurodegenerative disorders like Alzheimer’s disease. Its ability to modulate cellular defense mechanisms enhances its potential in age-related cognitive decline prevention.

In addition, Dehydroglyasperin C demonstrates antidiabetic activity by improving insulin sensitivity and glucose uptake in cell models, indicating possible use in managing type 2 diabetes. It also has antimicrobial and anticancer properties under investigation, where it has been observed to suppress the growth of certain cancer cell lines through induction of apoptosis and cell cycle arrest.

Due to its multifunctional bioactivity, Dehydroglyasperin C is considered a valuable natural compound for developing functional foods, dietary supplements, and pharmaceutical agents targeting metabolic, neurological, and inflammatory conditions.