1-(5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl)-N-methylmethanamine fumarate

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Reagent Code: #188128
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CAS Number 881681-01-2

science Other reagents with same CAS 881681-01-2

blur_circular Chemical Specifications

scatter_plot Molecular Information
Weight 461.46 g/mol
Formula C₂₁H₂₀FN₃O₆S
badge Registry Numbers
MDL Number MFCD18633280
inventory_2 Storage & Handling
Storage Store in an inert gas at room temperature

description Product Description

Used in pharmaceutical research as a potent and selective antagonist for serotonin receptors, particularly 5-HT6, showing potential in the development of cognitive enhancers for neurodegenerative disorders such as Alzheimer's disease. Demonstrates good blood-brain barrier penetration and oral bioavailability in preclinical models, making it a valuable candidate in studies targeting memory impairment and neurobehavioral conditions. Also employed in structure-activity relationship (SAR) studies to optimize receptor binding affinity and selectivity in central nervous system drug discovery.

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Size Availability Unit Price Quantity
inventory 100mg
10-20 days ฿143.00
inventory 1g
10-20 days ฿1,310.00
inventory 5g
10-20 days ฿2,513.50
inventory 250mg
10-20 days ฿490.00

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1-(5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl)-N-methylmethanamine fumarate
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Used in pharmaceutical research as a potent and selective antagonist for serotonin receptors, particularly 5-HT6, showing potential in the development of cognitive enhancers for neurodegenerative disorders such as Alzheimer's disease. Demonstrates good blood-brain barrier penetration and oral bioavailability in preclinical models, making it a valuable candidate in studies targeting memory impairment and neurobehavioral conditions. Also employed in structure-activity relationship (SAR) studies to optimize receptor binding affinity and selectivity in central nervous system drug discovery.
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