Used as a key intermediate in the synthesis of biologically active compounds, particularly in pharmaceutical research. It serves as a building block for kinase inhibitors and other nitrogen-containing heterocyclic systems. The iodine substituent at position 3 allows for further functionalization via cross-coupling reactions such as Suzuki or Heck couplings, enabling rapid diversification in drug discovery programs. The tert-butoxycarbonyl (Boc) group protects the nitrogen at position 1, helping to control reaction specificity and can be removed under mild acidic conditions. Commonly employed in the development of potential treatments for cancer, inflammation, and central nervous system disorders due to its role in constructing pyrazolopyridine scaffolds known for their pharmacological relevance.