Used as an intermediate in the synthesis of biologically active compounds, particularly in pharmaceutical research targeting kinase inhibitors. Its structure supports the development of chiral molecules with high stereoselectivity, making it valuable in the creation of potential antitumor and anti-inflammatory agents. The presence of the iodopyrazole moiety allows for further functionalization via cross-coupling reactions, enabling rapid diversification in drug discovery programs. Commonly employed in medicinal chemistry for building blocks in the development of targeted therapies.