7-Aminoflavone is primarily investigated for its potential biological and pharmacological applications. It exhibits notable anti-cancer properties by inhibiting specific kinases involved in tumor cell proliferation, making it a candidate for targeted cancer therapy. Research also highlights its role as a modulator of metabolic enzymes, particularly in detoxification pathways, which may contribute to chemopreventive strategies. Additionally, 7-aminoflavone shows anti-inflammatory and neuroprotective effects in preclinical models, suggesting possible use in treating neurodegenerative conditions such as Alzheimer’s disease. Its ability to cross the blood-brain barrier enhances its suitability for central nervous system-related therapeutic development. The compound is also used as a chemical intermediate in synthesizing more complex flavone derivatives with optimized bioactivity.