tert-Butyl (2-(1H-imidazol-5-yl)ethyl)carbamate is primarily used in organic synthesis and pharmaceutical research. It serves as a key intermediate in the development of various biologically active compounds, particularly those targeting enzyme inhibition or receptor modulation. The imidazole moiety in its structure makes it valuable for designing molecules with potential therapeutic applications, such as antifungal, antibacterial, or anticancer agents. Additionally, it is utilized in peptide chemistry for protecting amine groups during complex synthetic processes. Its stability and reactivity make it a versatile building block in medicinal chemistry and drug discovery.