Tigogenin is widely used in the pharmaceutical industry as a starting material for the synthesis of steroidal drugs. It serves as a key intermediate in the production of corticosteroids, sex hormones, and other therapeutic steroids. Its anti-inflammatory and cholesterol-lowering properties make it valuable in developing treatments for conditions like arthritis and cardiovascular diseases. Additionally, tigogenin is utilized in research to study its potential anticancer and neuroprotective effects. In traditional medicine, it is incorporated into formulations for its purported health benefits, such as improving liver function and boosting immunity. Its role in plant biochemistry also makes it a subject of interest in agricultural studies.