Linarin is widely studied for its anti-inflammatory and antioxidant properties, making it a promising compound in the development of natural therapeutic agents. It has shown potential in reducing neuroinflammation, which suggests possible applications in treating neurodegenerative disorders such as Alzheimer’s disease. Research also indicates that linarin exhibits sedative and anxiolytic effects, supporting its traditional use in promoting sleep and reducing anxiety. Due to its ability to modulate neurotransmitter systems like GABA, it may contribute to the formulation of herbal sedatives or sleep aids. Additionally, linarin has demonstrated hepatoprotective activity, helping protect liver cells from damage caused by toxins. Its presence in various medicinal plants makes it a valuable marker for quality control in herbal products. Ongoing studies explore its potential in managing diabetes and cancer, owing to its antihyperglycemic and cytotoxic effects in preclinical models.