Lithospermoside is a natural compound primarily used in skincare and cosmetic formulations for its multifaceted benefits. It exhibits anti-inflammatory and skin-soothing properties, helping to reduce redness and irritation, making it ideal for sensitive or reactive skin types. The compound supports the skin’s natural barrier function and is commonly included in products targeting conditions like eczema, dermatitis, or post-procedure recovery. Additionally, lithospermoside inhibits tyrosinase activity, reducing melanin production to help even skin tone, fade hyperpigmentation, dark spots, and freckles. Its potent antioxidant activity protects the skin from environmental stressors, including UV radiation and pollution, contributing to the prevention of premature aging and promoting a youthful appearance. In traditional medicine, extracts containing lithospermoside have been used to promote wound healing and treat minor skin injuries. It is often incorporated into sunscreens, serums, and restorative creams.