Isorhoifolin exhibits significant biological activities, making it valuable in pharmaceutical and cosmetic applications. It is studied for its anti-inflammatory properties, helping to reduce inflammation markers in cellular models. The compound also shows antioxidant effects, protecting cells from oxidative stress, which is beneficial in anti-aging formulations. In dermatology, Isorhoifolin is used to support skin health by improving elasticity and reducing irritation. Additionally, it has demonstrated potential in managing allergic responses due to its antihistaminic activity. Research explores its role in metabolic regulation, particularly in glucose uptake, suggesting possible applications in managing metabolic disorders. Its natural origin and low toxicity profile make it suitable for inclusion in nutraceuticals and functional foods aimed at promoting overall wellness.