Artemetin is primarily studied for its potential antimalarial properties, showing activity against Plasmodium species, including strains resistant to conventional drugs like chloroquine. It enhances the effectiveness of other antimalarial agents when used in combination therapies. Beyond malaria, artemetin exhibits anti-inflammatory and anticancer activities. It has demonstrated cytotoxic effects on various cancer cell lines by inducing apoptosis and inhibiting cell proliferation. Research also suggests antioxidant properties, which may contribute to its therapeutic effects in reducing oxidative stress-related damage. Due to its natural origin and bioactivity, artemetin is of interest in the development of phytopharmaceuticals and complementary medicine formulations.