Used as a potent selective antagonist for the GPR132 receptor, this compound is primarily applied in pharmacological research to study immune cell signaling and inflammatory processes. It helps modulate macrophage activity, making it valuable in investigating chronic inflammatory diseases, autoimmune disorders, and cancer-related inflammation. Due to its high selectivity and cellular permeability, it is also employed in target validation studies and early-stage drug discovery programs focused on G protein-coupled receptors. Its stability in biological assays allows for reliable in vitro and in vivo experimentation.