tert-Butyl (2-oxo-1,2-dihydropyridin-3-yl)carbamate is primarily used in organic synthesis and pharmaceutical research. It serves as a key intermediate in the development of various biologically active compounds, particularly in the synthesis of heterocyclic molecules. Its structure is valuable for constructing complex pharmacophores, often utilized in the design of drugs targeting neurological disorders, inflammation, and cancer. The compound is also employed in medicinal chemistry for the preparation of pyridine derivatives, which are essential in creating molecules with potential therapeutic applications. Additionally, it is used in the study of enzyme inhibition and receptor binding due to its ability to mimic certain natural substrates.