Used as a key intermediate in the synthesis of pharmaceutical agents, particularly in the development of central nervous system (CNS) active compounds. Its structure supports binding to neurological targets, making it valuable in creating drugs for psychiatric and neurological disorders. The amine functionality allows for easy derivatization, enabling the formation of amides, sulfonamides, or other conjugates to optimize drug potency and selectivity. Commonly employed in medicinal chemistry research for structure-activity relationship (SAR) studies due to its rigid tetrahydropyran core and lipophilic trifluoromethoxyphenyl group, which enhance blood-brain barrier penetration. Also utilized in the preparation of selective enzyme inhibitors and receptor modulators in preclinical drug discovery programs.