Probucoldisuccinate is the disuccinate salt of probucol, primarily utilized in the development of pharmaceutical formulations for managing hyperlipidemia. It works by promoting cholesterol efflux from cells and tissues, enhancing reverse cholesterol transport, and exhibiting antioxidant properties that help prevent LDL oxidation, thereby lowering cholesterol levels in the blood and reducing the risk of cardiovascular diseases. This compound is often incorporated into oral medications for patients with high cholesterol or at risk of atherosclerosis. Its anti-atherogenic effects make it a valuable component in lipid-lowering therapies. Research highlights its potential to protect cells from oxidative stress, further benefiting cardiovascular health. Probucoldisuccinate is formulated to ensure optimal bioavailability and efficacy in clinical applications.