6,7-Bis(benzyloxy)coumarin is primarily utilized in the field of organic synthesis and pharmaceutical research. It serves as a key intermediate in the development of various biologically active compounds, particularly those with potential therapeutic applications. The compound is often employed in the synthesis of coumarin derivatives, which are known for their diverse pharmacological properties, including anti-inflammatory, antioxidant, and anticancer activities. Additionally, it is used in the study of enzyme inhibition and as a fluorescent probe in biochemical assays due to its unique photophysical properties. Its benzyloxy groups make it a valuable precursor for further chemical modifications, enabling the creation of more complex molecules with specific biological targets.