Cerberic acid B is primarily studied for its potent biological activity, particularly in neuropharmacology. It acts as a selective modulator of GABA-A receptors, making it a valuable tool in neuroscience research for understanding inhibitory neurotransmission. Due to its ability to influence chloride ion channels associated with GABA receptors, it has been used experimentally to investigate anxiety, seizure disorders, and sleep regulation. Its high specificity allows researchers to probe receptor subtypes, aiding in the development of targeted central nervous system drugs. Additionally, cerberic acid B has shown cytotoxic effects in certain cancer cell lines, suggesting potential as a lead compound in oncology research, though this application remains in early stages.