Canophyllal is primarily used in organic synthesis as a key intermediate in the preparation of complex natural products and bioactive molecules. Its unique structural features make it valuable in the development of pharmaceuticals, particularly in the synthesis of compounds with potential anticancer and anti-inflammatory properties. It is also employed in fragrance chemistry due to its terpenoid backbone, contributing to the creation of natural-identical aroma compounds used in perfumery and flavoring. Additionally, Canophyllal serves as a chiral building block in asymmetric synthesis, enabling the construction of stereochemically defined molecules important in drug discovery.