6,8-Diprenylgenistein is a bioactive compound with potential applications as an active ingredient, particularly for its antioxidant properties, which help reduce cellular damage from oxidative stress. It also exhibits anti-inflammatory effects, which may be beneficial in developing treatments for chronic inflammatory conditions such as arthritis or metabolic disorders.

Some research has found that this compound has anti-proliferative effects on cancer cells, especially breast and colon cancer cells, making it interesting as a lead compound for future anti-cancer drug development. It also inhibits certain enzymes involved in cancer cell metastasis.

Due to its structure similar to flavonoids found in herbal plants, this substance may be used in dietary supplements or cosmetics to promote skin health and anti-aging. It is used in skincare formulations for its antioxidant and anti-aging properties, helping protect skin cells from oxidative stress and potentially supporting collagen production. It is found in anti-wrinkle creams and serums targeting fine lines and sun damage, and studied for anti-inflammatory effects in dermatological applications.