Artocarpin is a bioactive flavonoid primarily studied for its pharmacological properties. It exhibits strong anti-inflammatory and antioxidant activities, making it a candidate for use in treating chronic inflammatory conditions and oxidative stress-related diseases. Research suggests artocarpin can inhibit key enzymes involved in inflammation, such as cyclooxygenase and lipoxygenase, which may lead to its application in developing natural anti-arthritic or anti-allergic agents. Furthermore, it has been reported to inhibit alpha-glucosidase, an enzyme involved in carbohydrate digestion, potentially aiding in blood glucose control and suggesting applications in anti-diabetic formulations.

It has also shown potential in cancer research due to its ability to induce apoptosis and suppress proliferation in certain cancer cell lines, including those of the liver, breast, and colon. Its antimicrobial activity against a range of bacteria and fungi supports its traditional use in treating infections and opens possibilities for development in topical antimicrobial formulations.

Additionally, artocarpin has been investigated for its skin-protective effects, particularly in inhibiting melanin production, suggesting a role in cosmetic applications for managing hyperpigmentation and promoting skin lightening. Due to its natural origin and multi-target biological activities, it is considered a valuable compound in nutraceuticals, functional foods, and herbal medicine formulations.