Glochidiolide is primarily studied for its potential biological activities, particularly in the field of natural product-based drug discovery. It has shown promising cytotoxic effects against certain cancer cell lines, making it a subject of interest in anticancer research. Its structure, belonging to the class of sesquiterpene lactones, contributes to its ability to interact with cellular targets involved in inflammation and cell proliferation. Due to these properties, Glochidiolide is investigated for its use in developing chemotherapeutic agents. Additionally, it may exhibit antimicrobial and anti-inflammatory activities, supporting its role in pharmaceutical and biomedical applications. Research remains largely preclinical, focusing on mechanism of action and structural optimization for enhanced efficacy and reduced toxicity.