(R)-2-(Pyrrolidin-2-yl)acetic acid is utilized in the synthesis of various pharmaceutical compounds, particularly those targeting neurological and cardiovascular disorders. Its chiral structure makes it valuable in the development of enantiomerically pure drugs, enhancing their efficacy and reducing side effects. This compound serves as a key intermediate in the production of inhibitors for enzymes like DPP-4, which are crucial in managing type 2 diabetes. Additionally, it is employed in the creation of peptide-based therapeutics, where its pyrrolidine ring contributes to stabilizing secondary structures in peptides, improving their biological activity. In research, it is used to study receptor-ligand interactions, aiding in the discovery of new drugs for conditions such as hypertension and Alzheimer's disease. Its versatility also extends to agrochemicals, where it is incorporated into formulations designed to improve crop protection and yield.