GSK1324726A (I-BET726)

10mM in DMSO

Reagent Code: #190259
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CAS Number 1300031-52-0

blur_circular Chemical Specifications

scatter_plot Molecular Information
Weight 434.91 g/mol
Formula C₂₅H₂₃ClN₂O₃
badge Registry Numbers
MDL Number MFCD28144683
inventory_2 Storage & Handling
Storage -20°C

description Product Description

Used in research to modulate gene expression by inhibiting bromodomain-containing proteins, particularly BET family proteins. This compound shows potential in oncology studies due to its ability to suppress oncogenic transcription factors and disrupt cancer cell proliferation. It has been investigated in hematological malignancies and solid tumors for its anti-proliferative effects. Additionally, it is applied in epigenetic research to study chromatin remodeling and transcriptional regulation. Its selectivity makes it a valuable tool for probing BET protein functions in disease models.

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Size Availability Unit Price Quantity
inventory 1ml
10-20 days ฿8,470.00

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