N-Boc-Cyclopropylamine is widely used in organic synthesis as a versatile building block for the preparation of more complex molecules. It serves as a key intermediate in the synthesis of pharmaceuticals, particularly in the development of drugs targeting central nervous system disorders, cardiovascular diseases, and anti-inflammatory agents. Its cyclopropyl group is often incorporated into drug molecules to enhance metabolic stability and bioavailability. Additionally, it is utilized in peptide chemistry for the protection of amine groups during multi-step synthesis processes. Its role in creating chiral compounds and facilitating asymmetric synthesis further highlights its importance in medicinal chemistry and drug discovery.