Alpinumisoflavone acetate exhibits significant biological activity, making it valuable in pharmaceutical and biomedical research. It has demonstrated strong anti-inflammatory effects by inhibiting key inflammatory mediators such as nitric oxide and prostaglandins, suggesting potential use in treating chronic inflammatory diseases. The compound also shows promise as an anticancer agent, with studies indicating it can induce apoptosis and suppress proliferation in various cancer cell lines, including those of the breast, liver, and colon. Its ability to modulate signaling pathways like NF-κB and MAPK further supports its therapeutic potential. Additionally, alpinumisoflavone acetate possesses antimicrobial properties, effective against certain bacteria and fungi, which could lead to its application in developing new antimicrobial agents. Due to its natural origin and bioactivity, it is also explored in the formulation of nutraceuticals and cosmeceuticals for skin protection and anti-aging benefits.