Used in organic synthesis as an intermediate for pharmaceutical compounds, particularly in the development of bioactive molecules and receptor ligands. Its structure supports conjugation in medicinal chemistry, making it valuable in creating potential anticancer and anti-inflammatory agents. Commonly utilized in Suzuki and other cross-coupling reactions due to the iodine moiety, enabling the formation of biaryl derivatives. Also serves as a building block in the synthesis of kinase inhibitors and CNS-targeted drugs owing to the morpholine ring’s favorable pharmacokinetic properties.