Pitofenone is primarily used as an antispasmodic agent, particularly in the treatment of conditions involving smooth muscle spasms. It is often employed in urology to alleviate spasms in the urinary tract, providing relief from pain and discomfort associated with conditions such as kidney stones or urinary infections. Additionally, it is sometimes combined with other medications to enhance its efficacy in managing gastrointestinal spasms, helping to reduce symptoms like cramping and bloating. Its ability to relax smooth muscles makes it a valuable component in therapeutic regimens aimed at improving patient comfort and facilitating recovery in various medical scenarios.