Used in the synthesis of pharmaceutical agents, particularly as an intermediate in the development of central nervous system (CNS) active compounds. Its structure supports binding to benzodiazepine receptors, making it valuable in the creation of anxiolytic and anticonvulsant drugs. The chiral (R)-configuration is critical for biological activity, enabling selective interaction with target receptors. It is also explored in medicinal chemistry for optimizing drug potency and reducing side effects in neuroactive therapeutics.