Gamabufotalin is primarily utilized in medical research due to its potent biological activities. It has shown significant potential in cancer therapy, particularly in inducing apoptosis in various cancer cell lines. Studies suggest that it can inhibit the growth of tumors by targeting specific cellular pathways, making it a candidate for developing anti-cancer drugs. Additionally, it has been explored for its cardiotonic effects, which could be beneficial in treating certain heart conditions. Its ability to modulate immune responses also opens avenues for its use in immunotherapy. Researchers are actively investigating its mechanisms to harness its therapeutic properties effectively.