Lupeol acetate is widely studied for its anti-inflammatory and anticancer properties. It has shown potential in inhibiting the growth of various cancer cells, including those of the skin, prostate, and colon, by inducing apoptosis and suppressing tumor-promoting pathways. Due to its ability to modulate key signaling molecules like NF-κB and STAT3, it is considered a promising candidate for developing chemopreventive agents. It also exhibits skin-protective effects, making it useful in cosmetic and dermatological formulations aimed at reducing UV-induced damage and aging. Additionally, lupeol acetate has antimicrobial activity, which supports its use in formulations targeting bacterial and fungal infections. Its natural origin and low toxicity profile enhance its appeal in pharmaceutical and nutraceutical applications.