Toddalosin is primarily used in research settings for its biological activity, particularly in studies related to enzyme inhibition and cellular signaling pathways. It has shown potential as an anti-inflammatory agent due to its ability to modulate specific protein kinases involved in immune responses. Additionally, toddalosin is investigated for its antimicrobial properties, exhibiting activity against certain Gram-positive bacteria. Its role in apoptosis regulation makes it a compound of interest in cancer research, where it helps in understanding cell survival and death mechanisms. Due to its natural origin and structural complexity, it also serves as a lead compound in the development of synthetic analogs with improved pharmacological profiles.