Lobetyolin is primarily used in traditional medicine and modern herbal formulations due to its significant bioactive properties. It exhibits anti-inflammatory and immunomodulatory effects, making it valuable in managing respiratory conditions such as bronchitis and asthma. The compound also demonstrates neuroprotective potential, supporting its use in cognitive health supplements and research on neurodegenerative diseases like Alzheimer's. Additionally, lobetyolin has shown antimicrobial activity, contributing to its inclusion in natural remedies for infections. Its antioxidant properties are leveraged in anti-aging formulations and liver-protective agents, where it helps reduce oxidative stress. Ongoing studies explore its role in cancer therapy due to preliminary findings of antitumor activity.