Clerosterol glucoside is primarily studied for its potential bioactive properties, particularly in traditional and modern herbal medicine. It has been associated with anti-inflammatory and immunomodulatory effects, making it a compound of interest in formulations aimed at managing chronic inflammatory conditions. Research also suggests possible hepatoprotective activity, supporting its use in liver health supplements. Additionally, due to its structural similarity to plant sterols, it may contribute to cholesterol-lowering effects by interfering with dietary cholesterol absorption in the gut. The compound is often found in medicinal plants and is being explored for inclusion in nutraceuticals and functional foods targeting metabolic and immune health.