Chimaphilin is primarily used in traditional and herbal medicine due to its bioactive properties. It exhibits antimicrobial and anti-inflammatory activities, making it valuable in formulations aimed at treating skin infections and reducing inflammation. Research also suggests potential antioxidant effects, which contribute to cellular protection and may support the development of natural health products. Its presence in certain plant extracts is leveraged in cosmetic applications for soothing irritated skin and enhancing product efficacy. Ongoing studies explore its role in supporting urinary tract health, as it has been historically used in folk remedies for related conditions.