Apiopaeonoside is primarily studied for its potential anti-inflammatory and neuroprotective properties. It has shown activity in modulating pathways related to oxidative stress, making it a compound of interest in research on neurodegenerative conditions such as Alzheimer's and Parkinson’s disease. It may also contribute to hepatoprotective effects, supporting liver health by reducing damage caused by toxins. Due to its natural origin and bioactive profile, it is investigated as a candidate for developing herbal-based therapeutics, particularly in traditional medicine systems where the source plant is used for treating fever, pain, and nervous disorders. Its application remains mostly in the preclinical research stage, focusing on pharmacological evaluation and mechanism of action.