(S)-2-(Cyclohexylamino)propanoic acid is primarily used in the field of organic synthesis and pharmaceutical research. It serves as a chiral building block for the development of various biologically active compounds. Its stereochemistry makes it valuable in the synthesis of enantiomerically pure drugs, particularly those targeting neurological and cardiovascular diseases. Additionally, it is utilized in the preparation of peptidomimetics, which are compounds designed to mimic the structure and function of peptides, aiding in drug discovery and development. The compound is also explored in the study of enzyme inhibitors and receptor ligands, contributing to advancements in medicinal chemistry.