Serpentinine is primarily used in scientific research, particularly in the field of natural product chemistry and pharmacology. It has attracted interest due to its structural complexity and potential bioactivity. Studies have explored its effects on the central nervous system, showing possible sedative and anticonvulsant properties. It is also investigated for its interaction with various neurotransmitter receptors, which may provide insights into new therapeutic agents for neurological disorders. Due to its natural occurrence in certain plants, it serves as a marker compound in chemotaxonomic studies and in the authentication of herbal materials. Its use remains largely confined to laboratory and experimental settings, with no widespread clinical or industrial application to date.